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Pubblicazioni

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Rivista

Codice:

E060692

ISSN:

0223-5234

Dati Generali

Dati Generali

Pubblicazioni (47)

Ordina Pubblicazioni:

ascendente
decrescente

1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity

Articolo

1,3-Dioxolane-Based Ligands Incorporating a Lactam or Imide moiety: Structure-Affinity/Activity Relationship at alpha1–Adrenoceptor subtypes and at 5-HT1A Receptors

Articolo

2-[N-Alkyl(R-phenyl)-aminomethyl]-3-phenyl-7-trifluoromethylquinoxalines as anticancer agents inhibitors of folate enzymes

Articolo

7-Hydroxy-2-substituted-4-H-1-benzopyran-4-one derivatives as aldose reductase inhibitors: a SAR study

Articolo

A rational approach to the design of flavones as xanthine oxidase inhibitors

Articolo

Amphiphilic ion pairs of tobramycin with lipoamino acids

Articolo

Application of a post-docking procedure based on MM-PBSA and MM-GBSA on single and multiple protein conformations

Articolo

Aryl thiosemicarbazones for the treatment of trypanosomatidic infections

Articolo

Bifunctional compounds targeting both D2 and non-α7 nACh receptors: Design, synthesis and pharmacological characterization

Articolo

Computational analysis of ligand recognition sites of homo- andheteropentameric 5-HT3 receptors

Articolo

Correlation hetween adrenergic alpha-receptorantagonists of tetramine disulfidesand benzodioxanes classes

Articolo

Crassiflorone derivatives that inhibit Trypanosoma brucei glyceraldehyde-3-phosphate dehydrogenase (TbGAPDH) and Trypanosoma cruzi trypanothione reductase (TcTR) and display trypanocidal activity

Articolo

Discovery and development of novel salicylate synthase (MbtI) furanic inhibitors as antitubercular agents

Articolo

Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and genomics

Articolo

Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer

Articolo

Host dihydrofolate reductase (DHFR)-directed cycloguanil analogues endowed with activity against influenza virus and respiratory syncytial virus

Articolo

IDENTIFICATION OF PYRAZOLO-PIPERIDINONE DERIVATIVES TARGETING YAP-TEAD INTERFACE 3 AS ANTICANCER AGENTS THROUGH INTEGRATED VIRTUAL SCREENING AND MASS SPECTROMETRY PROTEOMICS

Articolo

Identification of 4-amino-2-Pyridones as new potent PCSK9 inhibitors: From phenotypic hit discovery to in vivo tolerability

Articolo

Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign

Articolo

Identification of non-ATP-competitive α-carboline inhibitors of the anaplastic lymphoma kinase

Articolo

Methoxylated 2'-hydroxychalcones as antiparasitic hit compounds

Articolo

Molecular properties of the adrenergic alpha-receptor6. - Optimum carbon chain-length between the inner nitrogenand the sulfur of tetramine disulfides

Articolo

Molecular properties of the adrenergic alpha-receptors.4.Topographical and structural differences betweentissue-specific binding sites as revealedby benextramine and analogues.

Articolo

Molecular requirements of the active sites of thecholinergic receptors XVII. 1,3-oxathiolane nucleus as a carrier of the active moeties

Articolo

Naphthalimido Derivatives as Antifolate Thymidylate Synthase Inhibitors

Articolo

New dimeric cGMP analogues reduce proliferation in three colon cancer cell lines

Articolo

Preparation and optimization of PIT solid lipid nanoparticles via statistical factorial design.

Articolo

Relationship between quantum-chemical descriptors of proton dissociation and experimental acidity contants of variously hydroxylated coumarins. Identification of the biologically active species for xanthine oxidase inhibition

Articolo

Resolution of the potent α1-adrenoreceptor antagonist 2-[[[2-(2,6-dimethoxyphenoxy)ethyl]amino]methyl]-1,4-benzoxathian (benoxathian)

Articolo

Scouting new sigma receptor ligands: Synthesis, pharmacological evaluation and molecular modeling of 1,3-dioxolane-based structures and derivatives

Articolo

Structural requirements for adrenergic alpha-receptorcovalent occupancy by chiral tetramine disulfides

Articolo

Structure-affinity/activity relationships of 1,4-dioxa-spiro[4.5]decane based ligands at α1 and 5-HT1A receptors

Articolo

Structure-guided optimization of 3-hydroxybenzoisoxazole derivatives as inhibitors of Aldo-keto reductase 1C3 (AKR1C3) to target prostate cancer

Articolo

Synthesis and activity of a new series of chalcones as aldose reductase inhibitors

Articolo

Synthesis and alpha blocking activity of some analogues of idazoxan

Articolo

Synthesis and alpha-blocl«ing activity of some cyclicand opened analogues of WB 4101 (-)

Articolo

Synthesis and antiplatelet activity of thioaryloxyacids analogues of clofibric acid

Articolo

Synthesis and structureeactivity relationship studies in serotonin 5-HT4 receptor ligands based on a benzo[de][2,6]naphthridine scaffold

Articolo

Synthesis of N-(5,7-diamino-3-phenyl-quinoxalin-2-yl)-3,4,5-substituted anilines and N-[4[(5,7-diamino-3-phenylquinoxalin-2-yl)amino]benzoyl]-l-glutamic acid diethyl ester: evaluation of in vitro anti-cancer and anti-folate activities

Articolo

Synthesis, biological evaluation and molecular modeling of 1-oxa-4-thiaspiro- and 1,4-dithiaspiro[4.5]decane derivatives as potent and selective 5-HT1A receptor agonists

Articolo

Synthesis, biological evaluation and molecular modeling of novel azaspiro dihydrotriazines as influenza virus inhibitors targeting the host factor dihydrofolate reductase (DHFR)

Articolo

Synthesis, characterization and in vitro evaluation of amphiphilic ion pairs of erythromycin and kanamycin antibiotics with liposaccharides

Articolo

Synthesis, characterization, crystallographic analysis, antifungal and genotoxic properties of some 1-methyl-1H-imidazoles

Articolo

Synthesis, chemical and biological studies on new Fe3þ-glycosilated b-diketo complexes for the treatment of iron deficiency

Articolo

The discovery of aryl-2-nitroethyl triamino pyrimidines as anti-Trypanosoma brucei agents

Articolo

Theoretical and experimental study of flavones as inhibitors of xanthine oxidase

Articolo

X-ray crystal structures of Enterococcus faecalis thymidylate synthase with folate binding site inhibitors

Articolo

No Results Found

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